Review on Biological Activities of 1,3,4-Thiadiazole Derivatives

Arvind k. Singh, Geeta Mishra, Kshitiz Jyoti

Pages: 44-49

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Design, Characterization and Biological Activity of a new series of s-Triazines Derived with Morpholine

Kalpesh S. Parikh, Sandip P. Vyas

DOI: 10.7324/JAPS.2012.2519Pages: 111-114

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Biological activities of [1,2,4] triazolo-[3,4-b],[1,3,4]-thiadiazole-6-yl) (o-tolyamino) methylazetidin-2-one

Harcharan Lal, Neeraj Sharma, T.P. Agarwal and Nitin Sharma

DOI: 10.7324/JAPS.2012.21021Pages: 104-112

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Solid Dispersion: Methods and Polymers to increase the solubility of poorly soluble drugs

Ladan Akbarpour Nikghalb, Gurinder Singh, Gaurav Singh and Kimia Fazaeli Kahkeshan

DOI: 10.7324/JAPS.2012.21031Pages: 170-175

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Molecular docking study of 3,6 bis(3’substituted propoxy) and 3,6 bis (5’substituted pentyloxy) xanthone derivatives as PGHS- 2 inhibitors

Aparoop Das, Pratap Parida, Neha Agarwal, Jaya shree, Brajesh Shankar and Dipankar Chakraborty

DOI: 10.7324/JAPS.2013.34.S3Pages: S13-S22

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Binding affinity of asiatic acid derivatives design against Inducible Nitric Oxide Synthase and ADMET Prediction

RE Kartasasmita, I Musfiroh, A Muhtadi, S Ibrahim

DOI: 10.7324/JAPS.2014.40213Pages: 075-080

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Design, synthesis, molecular docking of new thiopyrimidine-5-carbonitrile derivatives and their cytotoxic activity against HepG2 cell line

Ahmad F. Eweas, Qasem M.A. Abdallah, Emad S.I. Hassan

DOI: 10.7324/JAPS.2014.41218Pages: 102-111

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Synthesis of barbituric acid derivatives using microwave irradiation method and in vitro evaluation of antimicrobial and cytotoxic activity

M. A. Sattar, Mst. Khodeza Khatun, Rafiquel Islam, Md. Hossain Sohrab, Sharif M. Al-Reza

DOI: 10.7324/JAPS.2015.501106Pages: 038-042

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Recent Advances and Future Prospects of Phthalimide Derivatives

Neelottama Kushwaha, Darpan Kaushik

DOI: 10.7324/JAPS.2016.60330Pages: 159-171

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Pyrimidinethione derivatives with tosyl substitution: Synthesis, and antimicrobial property investigation

Shubhalaxmi, B. S. Manjunatha, K. Ananda, K. Subrahmanya Bhat

DOI: 10.7324/JAPS.2016.60613Pages: 073-078

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QSAR and Molecular Docking of Phthalazine Derivatives as Epidermal Growth Factor Receptor (EGFR) Inhibitors

Monika G. Shinde, Siddharth J. Modi, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2017.70427Pages: 181-191

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Design, Synthesis and Preliminary Pharmacological Screening (antimicrobial, analgesic and anti-inflammatory activity) of Some Novel Quinazoline Derivatives

Biswajit Dash, Suvakanta Dash, Damiki Laloo, Chitrani Medhi

DOI: 10.7324/JAPS.2017.70612Pages: 083-096

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Synthesis, Pharmacological Evaluation, Molecular Docking and in silico ADMET Prediction of Nitric Oxide Releasing Biphenyls as Anti-Inflammatory Agents

Monika G. Shinde, Siddharth J. Modi, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2017.71006Pages: 037-047

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Docking Evaluation of Catechin and its Derivatives on Fat Mass and Obesity-Associated (FTO) Protein for Anti-Obesity Agent

Tony Sumaryada, Renti Efraim Marimpola Simamora, Laksmi Ambarsari

DOI: 10.7324/JAPS.2018.8810Pages: 063-068

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The employment of spectroscopic techniques coupled with chemometrics for authentication analysis of halal pharmaceuticals

Abdul Rohman, Nina Salamah

DOI: 10.7324/JAPS.2018.81009Pages: 063-068

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3D-QSAR analysis of pyrimidine derivatives as AXL kinase inhibitors as anticancer agents

Siddharth J. Modi, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2018.81103Pages: 015-027

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Synthesis and anticancer potential of aminomethyl derivatives of methyl-substituted asymmetrical curcumin mono-carbonyl

Arini Kurnia, Fadlina Chany Saputri, Hayun Hayun

DOI: 10.7324/JAPS.2019.90803Pages: 018-024

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New benzimidazole derivatives as inhibitors of Pteridine reductase 1: Design, molecular docking study and ADMET prediction

Shraddha Phadke, Rakesh Somani, Devender Pathak

DOI: 10.7324/JAPS.2020.10904Pages: 030-039

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Design, synthesis, and evaluation of some novel N-benzothiazol-2-yl benzamide derivatives as allosteric activators of human glucokinase

Sandeep Arora, Ajmer Singh Grewal, Neelam Sharma, Kunal Arora, Ervon Dhalio, Sukhbir Singh

DOI: 10.7324/JAPS.2021.11s104Pages: 038-047

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Design, synthesis and in silico prediction of drug-likeness properties of new ortho, meta and para-(2-cyano-3-(3,5-di-tert-butyl-4- hydroxyphenyl)acrylamido)benzoic acids

Madhavi Kuchana, Lakshmi Bhavani Kambala

DOI: 10.7324/JAPS.2021.110805Pages: 031-035

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Evaluating the effect of amine-geldanamycin hybrids on anticancer activity

Tipparat Samsawat, Chanjira Jaramornburapong, Weerachai Phutdhawong, Waya S. Phutdhawong, Thongchai Taechowisan

DOI: 10.7324/JAPS.2021.110814Pages: 098-107

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Antioxidant potential and LC/MS metabolic profile of anticancer fractions from Echium angustifolium Mill. aerial parts

Hanan M. El-Tantawy, Ahmed R. Hassan, Hala E. Taha

DOI: 10.7324/JAPS.2021.1101220Pages: 200–208

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Synthesis and evaluation of novel 4-anilinocoumarin derivatives as potential antimicrobial agents

Sonia Yadav, Nitin Kumar, Vijay Bhalla

DOI: 10.7324/JAPS.2022.120518Pages: 196-204

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In silico and in vitro anti-cancer activity against breast cancer cell line MCF-7 of amide cinnamate derivatives

Teni Ernawati, Nina Artanti, Yudhi Dwi Kurniawan

DOI: 10.7324/JAPS.2024.162177Pages: 102-107

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Synthesis, in-vitro antioxidant and anti-inflammatory properties of novel amide derivatives of substituted 2-aminothiophenes and 3,4-dimethoxy cinnamic acid

Satya Sree Bandaru, Madhavi Kuchana

DOI: 10.7324/JAPS.2024.180925Pages: 116-125

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Scientific landscape of melatonin, its hybrids, and its derivatives as anti-tumor agents: A bibliometric analysis

Andres F. Yepes, Wilson Cardona Galeano, Howard Ramírez-Malule

DOI: 10.7324/JAPS.2024.169632Pages: 205-218

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Synthesis, in silico, and in vitro pharmacological evaluation of norbornenylpiperazine derivatives as potential ligands for nuclear hormone receptors

Karine Badalyan, Nelly Babayan, Elena Kalita, Narine Grigoryan, Natalya Sarkisyan, Ruzanna Grigoryan, Grigor Arakelov, Alexan Shahkhatuni, Hovhannes Attaryan, Davit Mkrtchyan, Hasmik Khachatryan, Lusine Khondkaryan

DOI: 10.7324/JAPS.2025.230239Pages: 115-127

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