Design, Synthesis and Preliminary Pharmacological Screening (antimicrobial, analgesic and anti-inflammatory activity) of Some Novel Quinazoline Derivatives

Biswajit Dash, Suvakanta Dash, Damiki Laloo, Chitrani Medhi

DOI: 10.7324/JAPS.2017.70612Pages: 083-096

Graphical Abstract

QSAR, Molecular Docking and Dynamics Studies of Quinazoline Derivatives as Inhibitor of Phosphatidylinositol 3-Kinase

Muhammad Arba, Ruslin, Waode Umi Kalsum, Armid Alroem, Muhammad Zakir Muzakkar, Ida Usman, Daryono Hadi Tjahjono

DOI: 10.7324/JAPS.2018.8501Pages: 001-009

Graphical Abstract

3D-QSAR, molecular docking, and dynamics simulation of quinazoline–phosphoramidate mustard conjugates as EGFR inhibitor

Ruslin Ruslin, Resky Amelia, Yamin Yamin, Sandra Megantara, Chun Wu, Muhammad Arba

DOI: 10.7324/JAPS.2019.90113Pages: 089-097

Graphical Abstract

Design, synthesis, and cytotoxicity evaluation of new 2,4-disubstituted quinazolines as potential anticancer agents

Gurubasavaraj V. Pujar, Syed Moshin Ali

DOI: 10.7324/JAPS.2020.10804Pages: 037-042

Graphical Abstract

Investigating the activity of Quinazoline derivatives against T790 mutant EGFR receptors employing computer-aided drug design

Deepika Dinesh Adottu, Afanamol Mankulathil Shajahan, Shifa Ali Koolaparambil, Shebina Pareed Rasheed, Ajeesh Vengamthodi, Suhail Pattilthodika, Arun Rasheed

DOI: 10.7324/JAPS.2024.188300Pages: 069-075

Graphical Abstract