Molecular Dynamic Simulation of Centella asiatica Compound as an Inhibitor of Advanced Glycation End Products
Lili Legiawati, Fadilah Fadilah, Kusmarinah Bramono, Siti Setiati, Em Yunir
DOI: 10.7324/JAPS.2020.10801Pages: 001-007
Microemulsion assisted transdermal delivery of a hydrophilic anti-osteoporotic drug: Formulation, in vivo pharmacokinetic studies, in vitro cell osteogenic activity
Mithila Boche, Varsha Pokharkar
DOI: 10.7324/JAPS.2020.10802Pages: 008-019
Design, synthesis, characterization, and cytotoxicity activity evaluation of mono-chalcones and new pyrazolines derivatives
Kassim Ali Salum, Mohammad Murwih Alidmat, Melati Khairulddean, Nik Nur Syazni Nik Mohammad Kamal, Musthahimah Muhammad
DOI: 10.7324/JAPS.2020.10803Pages: 020-036
Design, synthesis, and cytotoxicity evaluation of new 2,4-disubstituted quinazolines as potential anticancer agents
Gurubasavaraj V. Pujar, Syed Moshin Ali
DOI: 10.7324/JAPS.2020.10804Pages: 037-042
Evaluation of antidiabetic activities of Etlingera elatior flower aqueous extract in vitro and in vivo
Nor Asiah Muhamad Nor, Liza Noordin, Nor Hidayah Abu Bakar, Wan Amir Nizam Wan Ahmad
DOI: 10.7324/JAPS.2020.10805Pages: 043-051
Ethanolic extract of Moringa oleifera leaves improve inflammation, angiogenesis, and blood pressure in rat model of preeclampsia
Agnes Batmomolin, Ahsan Ahsan, I. Wayan Arsana Wiyasa, Sanarto Santoso
DOI: 10.7324/JAPS.2020.10806Pages: 052-057
Two novel antimicrobial and anticancer peptides prediction from Vibrio sp. strain ES25
Andis Sugrani, Ahyar Ahmad, Muhammad Natsir Djide, Hasnah Natsir
DOI: 10.7324/JAPS.2020.10807Pages: 058-066
Modulation impact of Diazinon forms on gene expression profile and DNA damage pathway in male mice
Neama I. Ali, Lamiaa M. Salem, Sawsan Y. Elateek, Wagdy K. B. Khalil
DOI: 10.7324/JAPS.2020.10808Pages: 067-074
A Schiff base of 2-((E)-(2-amino-5-methylphenylimino)methyl)- 5-(difluoromethoxy)phenol and its applications on fluorescent chemosensor for selection of Mg2+ ion, molecular docking, and anticancer activity
Iyappan Mathivanan, Dhineshkumar Ezhumalai, Anbuselvan Chinnadurai
DOI: 10.7324/JAPS.2020.10809Pages: 075-085
Passiflora ligularis leaf ultrasound-assisted extraction in the optimization of flavonoid content and enhancement of hypoglycemic activity
Paula M. Sepúlveda, Sandra Echeverrry, Geison Costa, Marcela Aragón
DOI: 10.7324/JAPS.2020.10810Pages: 086-094
Formulation and optimization of Enalapril Maleate-loaded floating microsphere using Box–Behnken design: in vitro study
Vijay Bahadur Kumal, Chhitij Thapa, Prakash Ghimire, Pradyumna Chaudhari, Jitendra Yadhav
DOI: 10.7324/JAPS.2020.10811Pages: 095-104
Thromboelastography as an instrument of preclinical studies of the potential drug
Aleksandr Livievich Urakov, Ilshat Ganeevich Mustafin, Rosa Mullayanovna Nabiullina, Linara Irekovna Bashirova, Konstantin Sergeevich Mochalov, Aleksandr Vladimirovich Samorodov, Ferkat Adelsyanovich Khaliullin, Danila Olegovich Lipatov, Vladislav Igorevich Korunas, Lina Nailevna Ismagilova, Almaz Radicovich Khalimov
DOI: 10.7324/JAPS.2020.10812Pages: 105-110
PCSK9 inhibitory activity of marine-derived compounds, aaptaminoids, and benzamide originated from Aaptos aaptos and Acanthaster planci as a potential treatment for atherosclerosis
Habsah Mohamad, Muhamad Fadzli Abd Razak, Nurjannatul Naim Kamaruddin, Lukman Hakim Mohd Din, Asnuzilawati Asari, Yosie Andriani, Siti Fatimah Zaharah Mustafa, Jasnizat Saidin, Muhammad Fadhlizil Fasihi Mohd Aluwi, Jalifah Latip, Tengku Sifzizul Tengku Muhammad
DOI: 10.7324/JAPS.2020.10813Pages: 111-123
High antibacterial properties of green synthesized gold nanoparticles using Uncaria gambir Roxb. leaf extract and triethanolamine
Syukri Arief, Fri Wardana Nasution, Zulhadjri, Arniati Labanni
DOI: 10.7324/JAPS.2020.10814Pages: 124-130
Simultaneous detection and quantification of bronchodilators in pure form and from in-vitro drug release of a novel combinational formulation
Sheena M. Raj, Vilas G. Jamakandi, Sunil S. Jalalpure, Pradeepkumar M. Ronad
DOI: 10.7324/JAPS.2020.10815Pages: 131-138
Molecular modeling, synthesis, and evaluation of 1-(4-methoxybenzofuran-5-yl)-3-phenylpropane-1, 3-dione for its anxiolytic potentiality
P Ayash Kumar, Sanjita Das, Sradhanjali Mohapatra, Saumya Priya Basu, Kalicharan Sharma, Monika Sharma, Aniruddh Pratap Singh
DOI: 10.7324/JAPS.2020.10816Pages: 139-144
Chelation activity and protective effect of Caulerpa lentillifera aqueous extract against lead acetate-induced toxicity in Sprague Dawley rats
Dzulsuhaimi Daud, Ahmad Nazrin Zainal, Muhammad Naqib Nordin, Alene Tawang, Asmida Ismail
DOI: 10.7324/JAPS.2020.10817Pages: 145-148
Chinese herbal medicine exhibits anticancer properties via eight cancer hallmarks
Menaga Subramaniam, Yang Mooi Lim
DOI: 10.7324/JAPS.2020.10818Pages: 149-163